Soluble guanylate cyclase as a direct target for pharmacologic mitigation of chronic kidney disease

Mia Jensen, Boye Lagerbon Jensen*

*Corresponding author for this work

Research output: Contribution to journalComment/debateResearchpeer-review

Abstract

In a preclinical rat study, Lichtenberger et al. show that BAY-60-2770, a drug that activates soluble guanylyl cyclase, often rendered inactive by oxidative stress, mitigates kidney inflammation, injury, and fibrosis, likely by vascular effects after ischemia-reperfusion. Kidney perfusion, overall vascular reactivity, and medullary microvascular diameter are improved by the drug at doses that do not alter blood pressure. Soluble guanylyl cyclase is an attractive and potentially unexploited target to halt progression of chronic kidney disease.

Original languageEnglish
JournalKidney International
Volume107
Issue number3
Pages (from-to)391-394
ISSN0085-2538
DOIs
Publication statusPublished - Mar 2025

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